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ENTRECTINIB CAP,ORAL

Clinical Criteria Summary

Exclusion Criteria

  • Prior history of prolonged QTc interval (repeated QTc interval >450 msec) or risk factors for torsade de pointes
  • Gastrointestinal condition that may interfere with entrectinib absorption
  • Interstitial lung disease, interstitial fibrosis, or tyrosine kinase inhibitor-induced pneumonitis
  • Prior ROS1 or NTRK tyrosine kinase inhibitor therapy
  • Unmanageable drug interaction identified
  • Creatinine clearance <30 mL/min
  • Total bilirubin >1.5 times the ULN (unless with Gilbert’s syndrome)
  • Pregnancy (i.e. known pregnancy or positive pregnancy test)
  • Breastfeeding

Inclusion Criteria

  • Care is provided by a VA/VA Community Care oncology provider
  • Eastern Cooperative Oncology Group (ECOG) performance status 0-2
  • Goals of care and role of Palliative Care consult have been discussed and documented
  • Female patients of child-bearing potential or male patients with female partner of child-bearing potential: counseling provided on contraception and risks vs. benefits of treatment; use effective contraception during therapy and for at least 5 weeks (female patients) or 3 months (males and female partners) after the final dose
  • Additional Inclusion Criteria (At least one must be met)
  • Patient with metastatic non-small cell lung cancer whose tumor is ROS1-positive
  • Patient with solid tumor that is metastatic or unresectable AND:
  • Has a neurotrophic tyrosine receptor kinase (NTRK) gene fusion without a known acquired resistance mutation AND
  • Has progressed following treatment or has no satisfactory alternative therapy

Source Documents