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ZOLBETUXIMAB-CLZB INJ,LYPHL

Clinical Criteria Summary

Document 729

Exclusion Criteria

  • PD-L1 by Combined Positive Score (CPS) > 5 (unless patient is not a candidate for an immune checkpoint inhibitor)
  • Prior severe allergic reaction or intolerance to known ingredients of zolbetuximab or other monoclonal antibodies, including humanized or chimeric antibodies
  • Absolute Neutrophil Count < 1500/mm3
  • Platelets < 100,000/mm3
  • Total bilirubin > 1.5x Upper Limit of Normal (or > 3x Upper Limit of Normal with liver metastases)
  • Estimated Creatinine Clearance < 30ml/min
  • Lactation

Inclusion Criteria

  • Locally advanced unresectable or metastatic gastric or gastroesophageal junction (GEJ) adenocarcinoma
  • HER2-negative tumor
  • CLDN18.2 positive tumor (≥75% of tumor cells showing moderate-to-strong staining)
  • Treatment plan includes zolbetuximab with a fluoropyrimidine- and platinum-based regimen (i.e. mFOLFOX6 or CAPOX) as first-line therapy
  • Care is provided by a VA/VA Community Care oncology or hematology provider
  • Eastern Cooperative Oncology Group (ECOG) performance status 0-2
  • Goals of care and role of Palliative Care consult have been discussed and documented

Additional Inclusion Criteria (if applicable)

  • For females who can become pregnant: Counseling provided on potential risks vs benefits of treatment; treatment should be given if the benefit outweighs the potential risk
  • For females who are lactating: breastfeeding/providing breastmilk to an infant is not recommended during therapy and for 8 months after stopping treatment.

Document 730

Indication & Patient Selection

  • First-line treatment of locally advanced unresectable or metastatic human epidermal growth factor receptor 2 (HER2) negative gastric or gastroesophageal junction adenocarcinoma
  • Tumors must be CLDN18.2 positive, as determined by an FDA-approved test
  • Administered in combination with fluoropyrimidine and platinum-containing chemotherapy (mFOLFOX6 or CAPOX)

Dosing & Administration

  • Initial dose: 800 mg/m2 IV
  • Subsequent doses: 600 mg/m2 IV every 3 weeks or 400 mg/m2 IV every 2 weeks
  • Continue therapy until disease progression or unacceptable toxicity
  • Supplied as 100 mg lyophilized powder in a single-dose vial

Monitoring & Safety Management

  • Monitor patients during the infusion and for 2 hours afterwards (or longer as needed) for hypersensitivity and infusion-related reactions
  • Pretreat patients with antiemetics prior to each infusion due to the highly emetogenic chemotherapy regimen
  • Manage nausea and vomiting with antiemetics, fluid replacement, infusion interruptions, and infusion rate adjustments

Clinical Pathway & Guideline Recommendations

  • NCCN Guidelines: Listed as a preferred first-line category 1 regimen for HER2-negative, CLDN18.2 positive locally advanced, unresectable, or metastatic gastric or GEJ cancer in combination with chemotherapy
  • VA Oncology Clinical Pathway (Esophageal Cancer V1.2025): Recommended first-line for stage IVB adenocarcinoma (HER2 negative, MSS) in patients who are candidates for cytotoxic chemotherapy, test positive for CLDN18.2, and are not candidates for immunotherapy or have PD-L1 CPS <5%

Source Documents